| Dr. | Abdo, Mohannad | Temptime Corporation | Technology Innovations Manager | Postdoctoral Associate | 2010 | Industry |  |
| Dr. | Abrous, Leila | California State... | Adjunct Professor of Chemistry and Biochemistry | Graduate Student | 1995 | Academia | |
| Dr. | Achab, Said | UniversitŽ de Reims,... | | Postdoc | | Academia | |
| Dr. | Adams, Chris | Novartis Pharmaceuticals... | Senior Investigator I | Graduate Student | 2003 | Industry | |
| Dr. | Adams, Greg | Merck | Senior Scientist | Graduate Student | 2008 | Industry |  |
| Dr. | Adams, Michael | US Food & Drug... | | | | Government | |
| Ai, Yanran | | | Graduate Student | 2009 | |  |
| Dr. | Akaishi, Ryouichi | Osaka Organic Chemical... | | Postdoc | | Industry | |
| Dr. | An, Chihui | Harvard University | Postdoctoral Fellow | Graduate Student | 2008 | |  |
| Dr. | Anand, Rajan | Merck & Co., Inc. | Research Scientist | Graduate Student | 1998 | Industry | |
| Dr. | Angeles, Angie | Merck-Boston | Associate Principal Scientist | Graduate Student | 2000 | Industry | |
| Prof. | Arimoto, Hirokazu | Tohoku University | Professor | | | Academia | |
| Arvary, Becky | Merck | Research Chemist | Masters | 2004 | Industry | |
| Dr. | Atasoylu, Onur | University of East Anglia | Independent Research Fellow in Medicinal Chemistry | Postdoctoral Associate | 2005 | N/A | |
| Dr. | Bacci, James | Provid Pharmaceuticals,... | Senior Research Scientist | Postdoctoral Associate | 2007 | Industry | |
| Dr. | Barbosa, Joseph | Lexicon Pharmaceuticals | Associate Director, Medicinal Chemistry | Graduate Student | 1998 | Industry | |
| Dr. | Basu, Kallol | Merck & Co., Inc. | Senior Scientist | | 2004 | Industry | |
| Dr. | Bauer, David | Amgen | Principal Scientist-Head of Med Chem outsourcing & Discovery Scale-Up | Postdoctoral Associate | 2001 | Industry | |
| Dr. | Beauchamp, Thomas | Eli Lilly & Company | Research Advisor | Graduate Student | 1998 | Industry | |
| Beiger, Jason | | | Undergrad | 2004 | | |
| Dr. | Belcher, Anne | | Retired | | | | |
| Benedetti, Phillip | The Boston Consulting... | Consultant | Masters | 2005 | Industry | |
| Prof. | Bennett, Clay | Tufts University | Assistant Professor | Graduate Student | 1999 | Academia | |
| Dr. | Benowitz, Andrew | GlaxoSmithKline | Senior Director | Graduate Student | 1993 | Industry | |
| Dr. | Bertounesque, Emmanuel | Institut Curie | Group Leader in Medicinal Chemistry | Postdoctoral Associate | 1991 | Academia | |
| Dr. | Beshore, Doug | Merck & Co., Inc. | Associate Principal Scientist | Graduate Student | 2004 | Industry | |
| Bezagu, Marine | | | | 2011 | |  |
| Prof. | Blase, Frances | Haverford College | Associate Professor | | | Academia | |
| Dr. | Bloom, Josh | American Council on... | Director of Chemical and Pharmaceutical Sciences | Postdoctoral Associate | | Industry | |
| Dr. | Boldi, Armen | Genentech | Senior Global Project Manager | Postdoctoral Associate | 1994 | | |
| Dr. | Bondar, Dmitriy | | | | 2005 | | |
| Dr. | Bosanac, Todd | Boehringer Ingelheim... | Principal Scientist | Postdoctoral Associate | 2003 | Industry | |
| Dr. | Boschelli, Diane | Parke-Davis | | Graduate Student | 1981 | Industry | |
| Dr. | Branca, Stephen | | Deceased | Graduate Student | 1978 | | |
| Dr. | Brandt, Benjamin | Johnson and Johnson | Patent Manager | Graduate Student | 2000 | Industry | |
| Dr. | Brard, Laurent | Woman and Infants... | | Postdoc | | Medicine | |
| Dr. | Brenneman, Jehrod | Boehringer Ingelheim | Principal Scientist | Postdoctoral Associate | 2005 | Industry | |
| Dr. | Brook, Chris | GlaxoSmithKline | Director | Postdoctoral Associate | 1994 | Industry | |
| Prof. | Brouard, Ignacio | University of La Laguna | | | 2003 | Academia | |
| Brown, Steve | | | Graduate Student | 2010 | |  |
| Dr. | Bunner, Matthew H. | Boehringer Ingelheim | Senior Scientist | Graduate Student | 2015 | Industry |  |
| Dr. | Byrne, Kevin | Seagrams, Inc. | | Postdoctoral Associate | | Industry | |
| Dr. | Cantin, Louis-David | Groupe PARIMA Inc. | Chief Scientific Officer | Postdoctoral Associate | 2001 | Industry | |
| Cattoen, Martin | | | Undergraduate Student, UPenn | 2014 | |  |
| Chanin, Jake | | | Undergraduate Student | 2005 | | |
| Chaplain, Cheyenne | MilliporeSigma | Senior Scientist | | | | |
| Dr. | Charnley, Adam | GlaxoSmithKline | Principal Scientist | Graduate Student | 2000 | Industry | |
| Dr. | Chen, Junhua | Exemplify Biopharma | Process Chemist | Postdoctoral Associate | 2017 | Industry |  |
| Dr. | Chen, Kwunmin | National Taiwan Normal... | Professor | Graduate Student | 1992 | Academia | |
| Dr. | Chen, Ming | Pfizer | Senior Scientist | Postdoctoral Associate | 2012 | Industry |  |
| Dr. | Chen, Shuyong | Bristol-Myers Squibb... | Sr. Research Investigator | Graduate Student | | Industry | |
| Dr. | Chida, Noritaka | Keio University | Professor of Chemistry | Postdoctoral Associate | 1988 | Academia | |
| Prof. | Cho, Cheon-Gyu | Hanyang University | Professor | | 2005 | Academia | |
| Dr. | Cho, Young Shin | Novartis Institutes for... | | Graduate Student | 2002 | Academia | |
| Dr. | Christie, Martin | Bettercoal | Executive Director | Postdoctoral Associate | 1988 | Industry | |
| Prof. | Chruma, Jason | Sichuan University... | Professor and Director of PhD Studies | Graduate Student | 2002 | Academia | |
| Dr. | Ciavarri, Jeff | Millenium Pharmceuticals | Research Chemist | Postdoctoral Associate | 2003 | Industry | |
| Dr. | Cichy-Knight, Maria | GlaxoSmithKline | Investigator | Graduate Student | 1998 | Industry | |
| Dr. | Clark, William | GlaxoSmithKline | Manager, Early Development Sciences, API Selection and Synthesis | | | Industry | |
| Dr. | Condon, Stephen | TetraLogic... | Vice President, Chemistry | Graduate Student | 1990 | Industry | |
| Dr. | Corbett, Mike | DuPont Crop Protection | Research Investigator | Graduate Student | 1999 | Industry | |
| Cornec, Anne-Sophie | | | Postdoctoral Associate | 2013 | |  |
| Dr. | Courter, Joel | jcourter@incyte.com | | Graduate Student | 2004 | Industry | |
| Cox, Joshua | MD Anderson Cancer Center | Medicinal Chemist | | | | |
| Dr. | Cox, Jason | Merck and Co.,Inc. | Research Fellow | | 2004 | Industry | |
| Dr. | Cui, Haifeng | GlaxoSmithKline | Chief Scientist | Graduate Student | 2002 | Industry | |
| Dr. | Davulcu, Akin | Bristol-Myers Squibb... | Senior Research Investigator | Graduate Student | 2003 | Industry | |
| Dr. | Degnan, Andrew | Bristol-Myers Squibb Co. | Principal Investigator | | 2002 | Industry | |
| Prof. | Dellinger, Barry | Louisiana State... | Patrick F. Taylor Chair of Environmental Chemistry | Postdoctoral Associate | 1976 | Academia | |
| Deng, Yifan | Gilead Sciences | Research Scientist | | | | |
| Dr. | Dible, Ben | | Patent Analyst | Postdoctoral Associate | 2009 | Academia | |
| Prof. | Dieter, Karl | Clemson University | Full Professor | Graduate Student | 1977 | Academia | |
| Doerksen, Rosalie | | | Undergraduate Student, UPenn | 2013 | | |
| Dr. | Dong, Shuzhi | Merck & Co. | Associate Principle Scientist | Postdoctoral Associate | 2007 | Academia | |
| Dr. | Donnelly, Joseph | Lockheed Corporation | | Postdoc | | Industry | |
| Dr. | Dormer, Peter | Merck & Co., Inc. | Associate Principle Scientist | Graduate Student | 1995 | Industry | |
| Dr. | Dorsey, Bruce | Teva | VP, Discovery Research | Graduate Student | 1987 | Industry | |
| Dr. | Dougherty, Victoria | Merck Sharp & Dohme... | | | 2001 | Industry | |
| Dr. | Duan, Jim Jing-Wu | Bristol-Myers Squibb | Research Fellow | Graduate Student | 1992 | Industry | |
| Dr. | Ducry, Laurent | Lonza Ltd. | Group Leader Bioconjugates R&D | Postdoctoral Associate | 2000 | Industry | |
| Dr. | Duffey, Matt | Michael Best &... | Patent Scientist | Postdoctoral Associate | 2006 | Industry | |
| Prof. | Dunlap, Norma | Middle Tennessee State... | Professor | | | Academia | |
| Dr. | Elban, Mark | GlaxoSmithKline | | Postdoctoral Associate | 2007 | Industry | |
| Prof. | Ellis-Davies, Graham | Mount Sinai School of... | Professor | | | Medicine | |
| Dr. | Empfield, James | Vertex Pharmaceuticals | VP, Chemistry and Drug Discovery | Graduate Student | 1985 | Industry | |
| Dr. | Falcone-Hindley, Margaret | Johnson & Johnson | Manager, R&D Quality and Compliance | Postdoctoral Associate | 1998 | Industry | |
| Farrell, Mark | | | Postdoctoral Associate | 2014 | |  |
| Dr. | Favor, David | Teva Pharmaceuticals | Research Scientist III | Graduate Student | 1993 | Industry | |
| Dr. | Fitch, Duke | Glaxo-SmithKline | Senior Counsel (Patents)/Investigator - Medicinal Chemistry | Undergraduate Student, UPenn | 1993 | Industry | |
| Dr. | Foister, Shane | Georgia Southern... | Visiting Faculty | | 2003 | Academia | |
| Dr. | Foley, Megan | Epizyme, Inc. | Sr. Scientist, Molecular Discovery | Graduate Student | 2002 | Industry | |
| Forestieri, Roberto | | | Postdoctoral Associate | 2014 | |  |
| Dr. | Fox, Richard | Bristol-Myers Squibb | Senior Research Investigator | Graduate Student | 2000 | Industry | |
| Dr. | Freeze, B. Scott | Millennium: The Takeda... | Scientist II, Medicinal Chemistry | Graduate Student | 2005 | Industry | |
| Dr. | Friedrich, Sarah | Bristol-Meyers Squibb... | | Graduate Student | 1999 | Industry | |
| Prof. | Friestad, Greg | University of Iowa | Associate Professor | Postdoctoral Associate | 1995 | Academia | |
| Dr. | Frohn, Michael | Amgen | Senior Scientist | | | Industry | |
| Dr. | Fruncillo, Rich | Richard Fruncillo MD PhD... | Owner | Undergraduate Student, UPenn | 1971 | Industry | |
| Prof. | Fuertes, Michael | Texas Tech University | Assistant Professor | Postdoctoral Associate | 2002 | Academia | |
| Dr. | Fujimoto, Katsumi | Sankyo Pharmaceutical... | Vice President | | | Industry | |
| Dr. | Fujiwara, Shinya | Chugai Pharmaceutical Cp... | Senior Researcher | Postdoc | | Industry | |
| Furuichi, Noriyuki | | | Postdoc | 2005 | | |
| Dr. | Gaffney, Althea | American Institute of Physics | Assistant Director of Student Programs | Graduate Student | 2015 | Academia |  |
| Dr. | Gallagher, Rex | | Private Consultant | | | Industry | |
| Dr. | Gallagher, William | Bristol-Myers Squibb | Senior Research investigator II | Postdoctoral Associate | 2003 | Industry | |
| Mr. | Garcia, Joshua | Campbell Alliance | Consultant | Graduate Student | 2007 | Industry | |
| Dr. | Gaunt, Matthew | University of Cambridge | Professor | Postdoctoral Associate | 1999 | Academia | |
| Dr. | Gay, Bryant | Upsher-Smith | Scientist I Preformulation | Postdoctoral Associate | 2012 | Industry |  |
| Dr. | Gladding, Jeff | Warner Babcock Institute... | Scientist | Graduate Student | 2004 | Industry | |
| Dr. | Gonzales, Stephen | University of Texas... | Senior Research Scientist | Graduate Student | 2007 | Industry |  |
| Dr. | Gotchev, Dimitar | Teva Pharmaceutical | Research Scientist | Postdoctoral Associate | 2003 | Industry | |
| Dr. | Gotoh, Hiroaki | Yokohama National... | Associate Professor | Visiting Scholar | | Academia | |
| Dr. | Green, Clive | AstraZeneca | Associate Director and Head of Sample Management | Postdoctoral Associate | 2000 | Industry | |
| Dr. | Grenier, Melissa | Glaxo Smith Kline | Research Scientist | Graduate Student | 2014 | Industry |  |
| Dr. | Guaciaro, Michael | SAI Life Sciences,Ltd. | Senior Director - Sales and Business Development | Graduate Student | 1977 | Industry | |
| Dr. | Guo, Boying | Johnson & Johnson | Scientist, Discovery Chemistry | Postdoctoral Associate | 2017 | Industry |  |
| Dr. | Guzman, Mark | Genentech | Technical Product Leader | Graduate Student | 1989 | Industry | |
| Prof. | Hale, Karl | Queen's University... | Professor of Organic and Medicinal Chemistry and Chemical Biology | Postdoctoral Associate | 1985 | Academia | |
| Dr. | Hall, Eric | Agriculture & Agri-... | | Postdoc | | Industry | |
| Dr. | Hamley, Peter | Sanofi | Global Head, External Research Opportunities and Sourcing LGCR | Postdoctoral Associate | 1991 | Industry | |
| Dr. | Han, Guoxia | University of... | | Postdoc | 2001 | Academia | |
| Han, Heeoon | | | Graduate Student | 2007 | |  |
| Dr. | Han, Qiang | Lexicon Pharmaceuticals | Research Scientist | Graduate Student | 2000 | Industry | |
| Dr. | Harada, Hironori | Astellas Research... | Associate Director | | 2003 | Academia | |
| Dr. | Hartz, Richard | Bristol-Myers Squibb | Principal Scientist | Graduate Student | 1996 | Industry | |
| Prof. | Haseltine, John | Kennesaw State University | Associate Professor | Graduate Student | 1988 | Academia | |
| Dr. | He, Ming | Wilmington Pharma Tech | | Postdoctoral Associate | 2008 | Industry |  |
| Higgins, Tyler | GSK | Investigator, Chemical Development | | | | |
| Prof. | Hirose, Tomoyasu | Kitasato University,... | Associate Professor | | 2003 | Academia | |
| Dr. | Hogan, Anne Marie | Warner Chilcott (Ireland... | Medicinal Chemist | | 2007 | Industry | |
| Hoye, Adam | Avid | | Postdoctoral Associate | 2010 | Industry |  |
| Dr. | Hrib, Nicholas | Hoechst Marion Roussel,... | | Postdoc | | | |
| Dr. | Hu, Liu | Amgen Inc. | | Postdoc | | Industry | |
| Huang, Longchuan | | | Postdoctoral Associate | 2011 | |  |
| Dr. | Hull, Ken | AstraZeneca R&D... | | Postdoc | | Industry | |
| Dr. | Huryn, Donna | Wyeth Research | Director | Graduate Student | 1986 | Industry | |
| Dr. | Hynes, John | Bristol-Myers Squibb | | Graduate Student | 1996 | Industry | |
| Dr. | Ishibashi, Hideaki | Nagoya University | | Graduate Student | 1996 | Academia | |
| Dr. | Ishikawa, Tomoyasu | Takeda Pharmaceutical... | Director of Medicinal Chemistry | | 2003 | Industry | |
| Dr. | Ishiyama, Haruaki | Ohu University | Associate Professor | Postdoctoral Associate | 1999 | Academia | |
| Dr. | Iwama, Seiji | Osaka City University | c/o Prof. Y. Ohfune | Postdoc | | Academia | |
| Dr. | Iwashima, Makoto | Astellas Pharma Inc. | Corporate Executive, Vice President of Research Planning & Administration | | | Industry | |
| Prof. | Jeon, Junha | University of Texas at... | Assistant Professor | | 2009 | Academia |  |
| Dr. | Johnson, David | Corixa | | Postdoc | | Industry | |
| Jones, David | Dow Agrosciences | Discovery Chemist | Postdoctoral Associate | 2010 | Industry |  |
| Dr. | Jones, David | 4iNNO, LLC | | Graduate Student | 1993 | Industry | |
| Prof. | Jonnalagadda, Subash | Rowan University | Assistant Professor | | 2005 | Academia | |
| Dr. | Jurica, Jon | | | Graduate Student | 2003 | | |
| Kanoh, Naoki | Tohoku University | Full Professor | Postdoctoral Associate | 1997 | Academia | |
| Dr. | Kaufman, Michael | Parke-David... | Research Chemist | Postdoc | | Industry | |
| Prof. | Kawasaki, Tomomi | Meiji Pharmaceutical... | Professor | | 1990 | Academia | |
| Dr. | Keenan, Terence | Helicon Therapeutics | | Postdoc | | Industry | |
| Dr. | Kellum, Alex | Pfizer | Staff Scientist | Graduate Student | 2014 | Industry | |
| Dr. | Kenesky, Craig S. | Wilson Sonsini Goodrich... | Patent Agent and Scientific Advisor | Graduate Student | 1990 | Patent Law | |
| Dr. | Kerns, Jeffrey | GlaxoSmithKline | Manager of Medicinal Chemistry | | | Industry | |
| PhD | Khartulyari, Anton | | | Postdoc | 2007 | Academia | |
| Dr. | Kikuchi, Osamu | Ube Industries, Ltd. | | Postdoc | 2003 | Industry | |
| Dr. | Kim, Dae-Shik | Eisai | Scientist | Graduate Student | 2002 | Industry | |
| Dr. | Kim, Won-Suk | MIT with Professor... | Postdoc | Graduate Student | 2005 | | |
| Dr. | Kinsho, Takeshi | Shin-Etsu Chemical Co.,... | | Postdoc | | Industry | |
| Kirk, Sharon | | | Postdoctoral Associate | 2016 | | |
| Dr. | Knight, Steve | GlaxoSmithKline | | Postdoc | | Industry | |
| Dr. | Kobayashi, Kaoru | ONO Pharmaceutical Co.,... | | Postdoc | | Industry | |
| Dr. | Kobayashi, Toyoharu | | | Postdoc | 2007 | Academia | |
| Prof. | Konopelski, Joseph | University of California... | | | | Academia | |
| Dr. | Koyanagi, Junichi | Josai University | | Postdoc | 2000 | Academia | |
| Dr. | Koziski, Kathleen | Rohm & Haas Co. | | Postdoc | | Industry | |
| Prof. | Kozmin, Sergey | University of Chicago | | Postdoc | | Academia | |
| Dr. | Kozystka, Mariya | ICL-IP America Inc. | Post Doctoral Scientist | Postdoctoral Associate | 2008 | Industry |  |
| Kurogi, Taichi | | | Graduate Student | 2014 | | |
| Prof. | Kürti, László | UT Dallas Southwest... | Assistant Professor | Graduate Student | 2006 | Academia | |
| Kutsumura, Noriki | | | Postdoc | 2007 | Academia | |
| Dr. | Laakso, Leif | Wyeth Research | | Graduate Student | 1997 | Industry | |
| Dr. | Labows, John | Colgate Palmolive, Inc. | | Postdoc | | Industry | |
| Dr. | LaMarche, Matthew | Millenium Pharmaceuticals | | Graduate Student | 2002 | Industry | |
| Lasfargeas, Caroline | | | Visiting Scholar | 2013 | | |
| Lassalas, Pierrik | | | Postdoctoral Associate | 2014 | |  |
| Dr. | Leahy, James | Exelixis Pharmaceuticals... | Director, Chemistry | Postdoc | | Industry | |
| Dr. | Leazer, John | Merck & Co. | | Graduate Student | 1995 | Industry | |
| Prof. | Lee, Dongjoo | | Assistant Professor | Graduate Student | 2001 | Academia | |
| Prof. | Leenay, Tamara | St. Cloud State... | Professor of Chemistry | Graduate Student | 1988 | Academia | |
| Dr. | Lender, Andreas | | | Postdoc | | Industry | |
| Li, Bo | | | Graduate Student | 2013 | |  |
| Ms. | Li, Ningkun | Harvard School of... | Dental Student | | 2010 | Academia | |
| Dr. | Lim, John | Yale University | | Undergraduate Student | | Academia | |
| Prof. | Lin, Li | Lanzhou University | Associate Professor | Visiting Scholar | 2014 | Academia |  |
| Dr. | Lin, Qiyan | Incyte Corporation | Sr. Principal Investigator | Graduate Student | 2000 | Industry | |
| Lippincott, Daniel | Actylis | Senior Chemist | | | | |
| Dr. | Liu, Hu | ImClone Systems Inc. | | Postdoc | | Industry | |
| Dr. | Liu, Jian | Merck & Co. | | Postdoc | | Industry | |
| Liu, Qi | | | Graduate Student | 2013 | |  |
| Dr. | Liverton, Nigel | Merck Research... | Chemistry Collaboration Lead, External Research | | | Industry | |
| Dr. | Lodise-Barbosa, Stephanie | BakerHostetler | Attorney | Graduate Student | 2000 | Industry | |
| Lou, Kevin | | | Undergraduate Student, UPenn | 2011 | |  |
| Dr. | Lupo, Andrew | Schering-Plough Research... | | Postdoc | | Industry | |
| Dr. | Maeda, Tetsuya | Yamanouchi... | | Postdoc | | Industry | |
| PhD | Maegawa, Tomohiro | Gifu Pharmaceutical... | Assistant Professor | Postdoc | 2007 | Academia | |
| Prof. | Maio, William | New Mexico State... | Assistant Professor | Postdoctoral Associate | 2008 | Academia | |
| Dr. | Malamas, Michael | Wyeth Research | | Graduate Student | 1984 | Industry | |
| Malamas, Patricia | FMC Corporation | | Graduate Student | 1983 | Industry | |
| Prof. | Maleczka, Robert | Michigan State University | Professor and Chair | | | Academia | |
| Mardjuki, Rachel | | | Undergraduate Student, UPenn | 2016 | | |
| Marotte, Antoine | | | Visiting Scholar | 2013 | | |
| Martinez-Solorio, Dionicio | | | | 2011 | |  |
| Dr. | McBriar, Mark | Schering-Plough Research... | | Graduate Student | 1999 | Academia | |
| Dr. | McCauley, John | Merck & Co., Inc. | Senior Research Fellow | Graduate Student | 1996 | Industry | |
| Dr. | McCauley, Jr., John | Zeneca Pharmaceuticals | | Postdoc | | Industry | |
| Dr. | McVaugh, Cheryl | University of California | Staff Scientist | Graduate Student | 2003 | Academia | |
| Meis, Regina | | | Graduate Student | 2002 | Industry | |
| Melillo, Bruno | | | Graduate Student | 2011 | |  |
| Melvin, Jason | | | Graduate Student | 2007 | |  |
| Dr. | Mesaros, Eugen | Cephalon, Inc. | | | 2002 | | |
| Dr. | Mewshaw, Richard | Wyeth Research | | Graduate Student | 1984 | Industry | |
| Dr. | Meyer, Emmanuel | | | Postdoc | 2003 | Academia | |
| Micikas, Bobby | N/A | N/A | | | | |
| Dr. | Miller-Sulikowski, Michelle | Vanderbilt University | enior Lecturer, Chemistry and Assoc. Director of Education, Vanderbilt Institute of Chemical Biology | Graduate Student | 1991 | Academia | |
| Prof. | Minakawa, Noriaki | The University of... | Professor | | 1995 | Academia | |
| Dr. | Minbiole, Kevin | Villanova University | Assistant Professor | Graduate Student | 2001 | Academia | |
| Dr. | Miura, Tomoya | Kyoto University | Senior Lecturer | Postdoctoral Associate | 2003 | Academia | |
| Dr. | Montgomery, Thomas | Duquesne University | Assistant Professor of Chemistry | Postdoctoral Associate | 2016 | | |
| Moraca, Francesca | | | Postdoctoral Associate | 2014 | | |
| Dr. | Moser, Bill | 3M Corporate Research... | Research Specialist | | | Industry | |
| Mowery, Brendan | | | Graduate Student | 2001 | | |
| Dr. | Murase, Noriaki | | Taisho Pharmaceutical Co., Ltd. | | | Industry | |
| Dr. | Myers, Michael | Bristol-Myers Squibb | Senior Research Investigator I | Postdoctoral Associate | 2006 | Industry | |
| Dr. | Nakayama, Kiyoshi | Daiichi Pharmaceutical... | | | | Industry | |
| Dr. | Neagu, Irina | Pharamacopeia, Inc. | | Postdoc | | Industry | |
| Dr. | Neelamkavil, Santhosh | | | | 2002 | | |
| Dr. | Nelson, Fran | Wyeth Research | | Graduate Student | 1992 | Industry | |
| Dr. | Ng, Danny | FibroGen, Inc. | Research Scientist, Medicinal Chemistry | | 2004 | Industry | |
| Nguyen, Minh | Stanford University | Postdoctoral Scholar | Graduate Student | | | |
| Nguyen, Minh | | | Graduate Student | 2011 | |  |
| Dr. | Nittoli, Thomas | Wyeth Research | | Postdoc | | Industry | |
| Dr. | Noda, Ichio | Astellas US Technologies... | Senior Director | | | Industry | |
| Prof. | Nolen, Ernest | Colgate University | Professor | | | Academia | |
| O'Brien, Kevin T. | Saul Ewing Arnstein & Lehr LLP | Patent Agent | | | | |
| Prof. | Ohba, Masashi | Kanazawa University | | Postdoc | | Academia | |
| Dr. | Ohmoto, Kazuyuki | Ono Pharmaceutical Co.,... | Director of Discovery Research Planning | | | Industry | |
| Dr. | Ohta, Mitsuaki | Astellas Pharma Inc. | Vice President | | | Industry | |
| Dr. | Ohtake, Hiro | Teikyo University | | | | Academia | |
| Dr. | Okano, Koji | Japan Tobacco Inc. | | Postdoc | | Industry | |
| Dr. | Okumura, Hiroyuki | Fujisawa Pharmaceutical... | Research Manager | Postdoc | | Industry | |
| Dr. | Onur, Atasoylu | Warner Chilcott | | Postdoctoral Associate | 2005 | Industry |  |
| Dr. | Orbin, Alia | Riverside Law | | Graduate Student | 2006 | Industry |  |
| Dr. | Ott, Greg | Teva Pharmaceuticals | Director, Medicinal Chemistry | Graduate Student | 1997 | Industry | |
| Oukoloff, Killian | | | Postdoctoral Associate | 2016 | | |
| Dr. | Paczkowski, Mark | Exxon | | Graduate Student | 1982 | Industry | |
| Pahil, Karanbir | | | Undergraduate Student, UPenn | 2014 | |  |
| Dr. | Paone, Dan | Merck & Co., Inc. | Medicinal Chemistry Team Lead | Graduate Student | 1998 | Industry | |
| Park, Jongwoo | | | Postdoctoral Associate | 2012 | | |
| Dr | Park, Jun | LG Chemical | Research Scientist | Postdoctoral Fellow | 2017 | Industry |  |
| Dr. | Pasternak, Alexander | Merck & Co., Inc. | Chemistry Program Team Lead | | | Industry | |
| Prof. | Peak, S. | Tulane University | Assistant Professor | Graduate Student | 1991 | Academia | |
| Dr. | Pedersen-Morris, Michelle | Pharmacopeia | | Postdoc | | Industry | |
| Prof. | Pérez Sestelo, José | University of Coruña | Professor | | 1994 | Academia | |
| Phillips, Barton | Oregon State University | | Graduate Student | 1998 | Academia | |
| PhD | Piscitelli, Francesco | | | Postdoc | 2009 | Academia | |
| Pitram, Suresh | Scripps Research... | Postdoc with K.B. Sharpless | Graduate Student | 1997 | Academia | |
| Dr. | Potuzak, Justin | Harvard | Research Scientist | | 2007 | Academia | |
| Dr. | Prasad, Vidya | Gilead | | Graduate Student | 2001 | Industry | |
| Qiu, Yuping | Bristol-Myers Squibb | | Graduate Student | 1997 | Industry | |
| Radtke, Mark Alexander | GSK | Investigator, Chemical Development | | | | |
| Dr. | Raheja, Neil | Ontogen Corporation | | Postdoc | | Industry | |
| Prof. | Rainier, Jon | University of Utah | | Postdoc | | Academia | |
| Dr. | Rano, Thomas | Janssen Pharmaceutical... | Principal Scientist | Graduate Student | 1989 | Industry | |
| Dr. | Razler, Thomas | Bristol-Myers Squibb... | Senior Research Investigator | Graduate Student | 2001 | Industry | |
| Dr. | Reichert, Janice | Tufts University/mAbs | Research Assistant Professor/Editor-in-Chief | Graduate Student | 1990 | Industry | |
| Dr. | Remiszewski, Stacy | Novartis Pharmaceuticals... | | Postdoc | | Industry | |
| Reznik, Samuel | | | Undergraduate Student | 2006 | Academia | |
| Dr. | Richards, Lauren | Du Pont - Merck... | | Postdoc | | Industry | |
| Prof. | Riera, Antoni | Universitat de Barcelona | | Postdoc | | Academia | |
| Dr. | Risatti, Christina | Bristol-Meyers Squibb... | Research Scientist II | | 2005 | Industry | |
| Dr. | Rivero, Ralph | GlaxoSmithKline | | Graduate Student | 1987 | Industry | |
| Prof. | Rizzo, Carmelo | Vanderbilt University | | Graduate Student | 1990 | Academia | |
| Robinson, D.J. | Incyte Genomics | | Graduate Student | 1995 | Industry | |
| Dr. | Rucker, Paul | Novartis Pharmaceuticals... | Research Investigator, II | | 2002 | Industry | |
| Ryu, Ki Moon | | | Graduate Student | 2007 | Academia | |
| Dr. | Safonov, Igor | GlaxoSmithKline | | Graduate Student | 2001 | Industry | |
| Prof. | Sakamoto, Satoshi | Tokyo Institute of... | Assistant Professor | | 2003 | Academia | |
| Dr. | Sakamoto, Yasuharu | RIKEN | Senior Research Scientist | Postdoctoral Associate | 2000 | Industry | |
| Prof. | Salvatore, Brian | Louisiana State... | Associate Professor | Graduate Student | 1993 | Academia | |
| Sanchez, Luis | | | | 2011 | |  |
| Dr. | Sasho, Setsuya | Kyowa Hakko Kogyo Co. | | Postdoc | | Industry | |
| Dr. | Saunders, Jeffrey | Agios Pharmaceuticals | VP Chemistry | | 1985 | Industry | |
| Dr. | Savinov, Sergey | | | | | Academia | |
| Dr. | Scarborough, Jr., Robert | COR Therapeutics, Inc. | | Graduate Student | 1979 | Industry | |
| Dr. | Schelhaas, Michael | Bayger AG | | Postdoc | | Industry | |
| Sfouggatakis, Chris | | | Graduate Student | 1999 | | |
| Dr. | Shakespeare, William | ARIAD Pharmaceuticals,... | Vice President, Drug Discovery | | | Industry | |
| Dr. | Shaw, Scott | Bristol-Myers Squibb | Sr. Research Investigator | Postdoctoral Associate | | Industry | |
| Dr. | Shimokawa, Ken'ichiro | Astellas Venture... | Investment Director | Graduate Student | 1995 | Industry | |
| Prof. | Shirai, Ryuichi | The University of Tokyo | | Postdoc | | Academia | |
| Dr. | Shirakami, Shohei | Astellas Pharma Inc. | Senior Researcher, Medicinal Chemistry I | | 2003 | Industry | |
| Dr. | Shvartsbart, Artem | Incyte | Discovery Chemistry | Graduate Student | 2009 | Industry |  |
| Dr. | Simov, Vladimir | Merck & Co., Inc. | Senior Research Scientist | Graduate Student | 2003 | Industry | |
| Dr. | Sivaramakrishnan, Hariharan | Hikal Ltd. | Vice President | Postdoc | | Industry | |
| Dr. | Slade, Joel | Ciba-Geigy Corp. | | Postdoc | | Industry | |
| Smith, David | | | | 2013 | | |
| Dr. | Smits, Helmars | | | Postdoc | 2007 | Academia | |
| Sobukawa, Masao | Tanabe Seiyaku, Co., Ltd. | | Postdoc | | Industry | |
| Dr. | Sokolsky, Alexander (Sasha) | Incyte Corporation | Research Investigator I | Graduate Student | 2010 | Industry |  |
| Spafford, Matt | | | Graduate Student | 2009 | |  |
| Dr. | Sperry, Jeff | Pfizer, Inc. | Senior Scientist | | | Industry | |
| Dr. | Spoors, Grant | GlaxoSmithKline | | Postdoc | | Industry | |
| Dr. | Sprengeler, Paul | Celera | | Postdoc | | Industry | |
| Prof. | Strongin, Robert | Louisiana State... | | Graduate Student | 1995 | Academia | |
| Suennemann, Hans | | | Postdoc | 2006 | Academia | |
| Dr. | Sugasawa, Keizo | Astellas Pharm Inc | Research Fellow | Postdoc | 2009 | Industry | |
| PhD | Sugawara, Akihiro | | | Postdoc | 2008 | Academia | |
| Sugiyama, Shimpei | | | | 2011 | |  |
| Prof. | Sulikowski, Gary | Texas A&M University | | Graduate Student | 1989 | Academia | |
| Sun, Alexander | | | | 2009 | |  |
| Dr. | Sunazuka, Toshiaki | Kitasato University... | Professor | Postdoctoral Associate | 1988 | Academia | |
| Dr. | Takahiro, Soeta | | | Postdoc | 2007 | Academia | |
| Dr. | Takeuchi, Makoto | Astellas Pharma Inc. | Corporate Executive, Vice President of Project Management | | 2002 | Industry | |
| Prof. | Taylor, Carol | Massey University | Associate Professor | Graduate Student | 1993 | Academia | |
| Dr. | Taylor, Michael | Parke Davis | | Postdoc | | Industry | |
| Tellis, John | | | Visiting Scholar | 2012 | | |
| Dr. | Thompson, Andrew | J-Star Research | President | Graduate Student | 1985 | Industry | |
| Dr. | Toder, Bruce | University of Rochester | | Graduate Student | 1981 | Academia | |
| Dr. | Tokuyama, Hidetoshi | Tohoku University | Professor | | | Academia | |
| Tomoika, Takashi | | | Postdoc | 2004 | | |
| Tong, Rongbiao | The Hong Kong University... | | Postdoctoral Associate | 2008 | Academia |  |
| Dr. | Trumper, Peter | Esertap Consultants | | Postdoc | | Industry | |
| Dr. | Tu, Chin-Yun | Wyeth Research | Section Manager - SG6 | Postdoc | | Industry | |
| Udal, Robert | | | Postdoc | 2002 | | |
| Dr. | Vaccaro, Hank | Schering-Plough Research... | | Graduate Student | 1989 | Industry | |
| Dr. | van Rijn, Rachel | N.V. Organon | | Graduate Student | 2000 | Industry | |
| Vanecko, John | | | Postdoc | 2003 | | |
| Venkatasa, Somisetti | | | Visiting Scholar | 2017 | | |
| Dr. | Verhoest, Patrick | Pfizer | | Graduate Student | 2001 | Industry | |
| Vijayendran, Krishna | | | Graduate Student | 2014 | | |
| Dr. | Visnick, Mike | Reata Pharmaceuticals | V.P. Medicinal Chemistry | | | Industry | |
| Walsh, Shawn | Merck | | Graduate Student | 1999 | Industry | |
| Dr. | Wan, Zehong | Neuroexcitation... | Director, Head of Chemistry | Graduate Student | 2000 | Industry | |
| Dr. | Wang, Wenyong | GlaxoSmithKline | | Graduate Student | 2001 | Industry | |
| Wang, Xiaozhao | | | | 2010 | |  |
| Weatherly, Cale | | | Postdoctoral Associate | 2015 | | |
| Dr. | Wellington, Judith | Clay Center for the Arts... | President & CEO | | | Industry | |
| Wendler, DJ | | | Graduate Student | 2014 | | |
| Dr. | Wexler, Barry | Bristol-Myers Squibb | | Graduate Student | 1982 | Industry | |
| Dr. | Wexler, Ruth | Bristol-Myers Squibb R... | Executive Director | Graduate Student | 1982 | Industry | |
| Williams, Brett | | | Graduate Student | 2008 | |  |
| Williams, Doug | | | Graduate Student | | | |
| Windisch, Vincent | Absorption Systems | Vice President | Graduate Student | 1988 | | |
| Dr. | Winzenberg, Kevin | CSIRO Materials Science... | Senior Principal Research Scientist,Flexible Electronics | Postdoctoral Associate | 1983 | Industry | |
| Dr. | Witherington, Jason | GlaxoSmithKline | Director & Head of Epi-Readers; Epinova DPU | | | Industry | |
| Dr. | Wong, Weichyun | SCI Pharmtech, Inc. | President | Graduate Student | 1993 | Industry | |
| Dr. | Wood, Jill | | | Graduate Student | 1991 | | |
| Prof. | Wood, John | Colorado State University | A.I. Meyers Professor of Chemistry | Graduate Student | 1991 | Academia | |
| Dr. | Wovkulich, Peter | Hoffmann-LaRoche, Inc. | | Postdoc | | Industry | |
| Wu, Andrew | | | Postdoc | 2005 | | |
| Prof. | Wuest, William | Temple University. | Assistant Professor | Graduate Student | 2003 | Academia | |
| Prof. | Xian, Ming | Washington State... | Associate Professor | | 2003 | Academia | |
| Xiangqin Li | | | Postdoctoral Associate | 2017 | |  |
| Xiong, Hui | | | Postdoc | 2005 | | |
| Dr. | Yager, Kraig | Celltech R&D, Inc. | | Postdoc | | Industry | |
| Dr. | Yanagisawa, Isao | Institute for Drug... | Director | Postdoc | | Industry | |
| Yang, Yun | | | Visiting Scholar | 2017 | | |
| Dr. | Yao, Wenqing | Incyte Corporation | SVP, Discovery Chemistry | Graduate Student | 1997 | Industry | |
| Dr. | Yarger, Ronald | Nabisco Foods Group | | Postdoc | | Industry | |
| Dr. | Yokoyama, Yasushi | Yokohama National... | Professor of Chemistry, Member of Research & Education Council, Vice-Dean of Graduate School of Engineering | Postdoctoral Associate | 1985 | Academia | |
| Dr. | Zawacki, Lisa | Pharmacopeia Inc. | | Postdoctoral Associate | | Industry | |
| Dr. | Zhang, Deyi | US Food and Drug... | Science Staff | Postdoctoral Associate | 1998 | Industry | |
| Dr. | Zhang, Nan | Scripps | Research Assistant | Graduate Student | 2014 | |  |
| Dr. | Zhang, Yiwen | Northwest A&F University | Tenure-Track Professor | Postdoctoral Associate | 2017 | Academia |  |
| Dr. | Zheng, Junying | Merck Research Laboratory | Associate Principal Scientist | Graduate Student | 2003 | Industry | |
| Zhu, Wenyu | Incyte Genomics | | Graduate Student | 2003 | Industry | |
| Dr. | Zhuang, Linghang | Vitae Pharmaceuticals | Director, Medicinal Chemistry | Graduate Student | 1998 | Industry | |
| Dr. | Zhuqing, Liu | Merck Sharp & Dohme | Senior Scientist | | 2007 | Industry | |
| Dr. | Zibuck, Regina | Wayne State University | Director of Undergraduate Studies | Graduate Student | 1986 | Academia | |
| Dr. | Zou, Yike | University of California, Los Angeles | Postdoctoral Fellow | Graduate Student | 2013 | Academia |  |
